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AI-driven high-throughput droplet screening of cell-free gene expression
期刊论文
NATURE COMMUNICATIONS, 2025
作者:
Zhu, Jiawei
;
Meng, Yaru
;
Gao, Wenli
;
Yang, Shuo
;
Zhu, Wenjie
Adobe PDF(2626Kb)
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收藏
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浏览/下载:351/5
|
提交时间:2024/07/26
high-throughput screening
droplet microfluidics
cell-free gene expression
artificial intelligence
synthetic biology
Inhibitor Development for α‑Synuclein Fibril's Disordered Region to Alleviate Parkinson's Disease Pathology
期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 卷号: 146, 期号: 41, 页码: 28282-28295
作者:
Zhang, Shenqing
;
Xiang, Huaijiang
;
Tao, Youqi
;
Li, Juan
;
Zeng, Shuyi
Adobe PDF(12245Kb)
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收藏
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浏览/下载:361/12
|
提交时间:2024/09/27
Neurodegenerative diseases
Nuclear magnetic resonance spectroscopy
Targeted drug delivery
Amyloid fibril
Disordered regions
EM techniques
High throughput screening
Intrinsically disordered regions
Membrane receptors
Pathological effects
Solid state NMR
Structure-activity relationships
α-synuclein
Selection of Leptin Surrogates by a General Phenotypic Screening Method for Receptor Agonists
期刊论文
BIOMOLECULES, 2024, 卷号: 14, 期号: 4
作者:
Wang T(王涛)
;
Xixi Chen
;
Guang Yang
;
Xiaojie Shi
Adobe PDF(1762Kb)
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浏览/下载:513/57
|
提交时间:2024/04/28
phenotypic screening
high-throughput screening
cytokine surrogate
receptor agonist
biological receptor activation-dependent cell survival (BRADS)
Discovery of a novel OGT inhibitor through high-throughput screening based on Homogeneous Time-Resolved Fluorescence (HTRF)
期刊论文
BIOORGANIC CHEMISTRY, 2023, 卷号: 139
作者:
Wu, Xinyu
;
Wang, Mingchen
;
Cao, Yu
;
Xu, Ying
;
Yang, Ziqun
Adobe PDF(12244Kb)
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收藏
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浏览/下载:265/1
|
提交时间:2024/03/03
O-GlcNAcylation
O-GlcNAc transferase
High-throughput screening
Inhibitor
Accelerated Design of Ultra-High-Performance Aramid Copolymers via a High-Throughput Screening Approach
期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2023, 卷号: 15, 期号: 34, 页码: 40877-40886
作者:
Yoo, Hyeonsuk
;
Muthoka, Ruth M.
;
Zhang, Xiangyu
Adobe PDF(7138Kb)
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收藏
|
浏览/下载:208/1
|
提交时间:2023/09/08
aramid copolymer
high-throughput screening
molecular dynamics simulation
topological data analysis
tensile strength
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors
期刊论文
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1
作者:
Zang, Yi
;
Su, Mingbo
;
Wang, Qingxing
;
Cheng, Xi
;
Zhang, Wenru
Adobe PDF(2374Kb)
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收藏
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浏览/下载:770/153
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提交时间:2023/03/10
high-throughput screening
SARS
CoV-2
main
papain-like
proteases
Discovery and characterization of a novel cGAS covalent inhibitor for the treatment of inflammatory bowel disease
期刊论文
ACTA PHARMACOLOGICA SINICA, 2022
作者:
Song, Jia
;
Yang, Rui-rui
;
Chang, Jie
;
Liu, Ya-dan
;
Lu, Cheng-hao
Adobe PDF(2708Kb)
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收藏
|
浏览/下载:415/0
|
提交时间:2022/10/27
cyclic GMP-AMP synthase
covalent inhibitor
inflammatory bowel disease
high-throughput screening
Molecular docking-based computational platform for high-throughput virtual screening
期刊论文
CCF TRANSACTIONS ON HIGH PERFORMANCE COMPUTING, 2022, 卷号: 4, 期号: 1, 页码: 63-74
作者:
Zhang, Baohua
;
Li, Hui
;
Yu, Kunqian
;
Jin, Zhong
Adobe PDF(969Kb)
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收藏
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浏览/下载:818/334
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提交时间:2022/10/14
Binding energy
Molecular modeling
Visualization
Web services
Websites
Active compounds
Computational platforms
Computer aided drug design
High-throughput
Large-scale computing
Molecular docking
Structure-based
Supercomputing
Ultra-large-scale computing
Virtual Screening
BARCODED COMBINATORIAL SCREENING FOR HIGHLY EFFICIENT OPTIMIZATION OF CELL-FREE PROTEIN SYNTHESIS SYSTEMS IN DROPLETS
会议论文
MICROTAS 2022 - 26TH INTERNATIONAL CONFERENCE ON MINIATURIZED SYSTEMS FOR CHEMISTRY AND LIFE SCIENCES, Hybrid, Hangzhou, China, October 23, 2022 - October 27, 2022
作者:
Zhu, Jiawei
;
Meng, Yaru
;
Ma, Conghui
;
Li, Jian
;
Liu, Yifan
收藏
|
浏览/下载:220/0
|
提交时间:2023/11/24
Bar codes
Biosynthesis
Cells
Cytology
Fluorescence
Proteins
Cell free protein synthesis
Combinatorial screenings
Droplet microfluidics
Efficient optimisation
Fluorescent barcode
High throughput screening
Massively parallels
Optimal conditions
Reaction conditions
Ultra-high
High-Throughput Screening Campaign Identified a Potential Small Molecule RXFP3/4 Agonist
期刊论文
MOLECULES, 2021, 卷号: 26, 期号: 24
作者:
Lin, Guangyao
;
Feng, Yang
;
Cai, Xiaoqing
;
Zhou, Caihong
;
Shao, Lijun
Adobe PDF(2352Kb)
|
收藏
|
浏览/下载:400/0
|
提交时间:2022/01/10
RXFP3
RXFP4
high-throughput screening
agonist
WNN0109-C011
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