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Discovery of novel GluN1/GluN3A NMDA receptor inhibitors using a deep learning-based method
期刊论文
ACTA PHARMACOLOGICA SINICA, 2025
作者:
Wang, Shi-hang
;
Zeng, Yue
;
Yang, Hao
;
Tian, Si-yuan
;
Zhou, Yong-qi
Adobe PDF(2216Kb)
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收藏
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浏览/下载:8/1
|
提交时间:2025/05/20
N
-methyl-
D
-aspartate receptors
GluN1/GluN3A
ligand-based virtual screening
scaffold hopping
deep learning
GeminiMol
Elucidating Contributions of Drug Transporters/Enzyme to Nonlinear Pharmacokinetics of Grazoprevir by PBPK Modeling With a Cluster Gauss-Newton Method
期刊论文
CPT-PHARMACOMETRICS & SYSTEMS PHARMACOLOGY, 2025
作者:
Yoshikado, Takashi
;
Aoki, Yasunori
;
Nakamura, Ryo
;
Shida, Saeko
;
Sugiyama, Yuichi
Adobe PDF(1329Kb)
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浏览/下载:94/3
|
提交时间:2025/02/17
CYP3A
Michaelis constant
middle-out approach
nonlinear pharmacokinetics
OATP1B
PBPK modeling
P-gp
Developing safe and efficient CGBE editor based on Cas-embedding strategy
期刊论文
SYNTHETIC AND SYSTEMS BIOTECHNOLOGY, 2025, 卷号: 10, 期号: 2
作者:
Lin, Tian
;
Wang, Xin
;
Zhang, Yu
;
Li, Guanglei
;
Huang, Xingxu
Adobe PDF(4784Kb)
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浏览/下载:70/2
|
提交时间:2025/03/03
CGBE
Cas-embedding
Off-target
eA3A
Regulation of de novo and maintenance DNA methylation by DNA methyltransferases in post-implantation embryos
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2024, 卷号: 301, 期号: 1
作者:
Xu, Zhen
;
Shi, Jiajia
;
Chen, Qian
;
Yang, Shuting
;
Wang, Zilin
Adobe PDF(1280Kb)
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浏览/下载:236/10
|
提交时间:2024/12/02
Cell culture
Gene encoding
Genome
Methylation
Stem cells
Bisulfite-sequencing
Control region
De novo methylation
DNA Methylation
DNMT1
DNMT3A
DNMT3B
Genomic imprinting
Implantation
Imprinting control region
Maintenance methylation
Whole-genome bisulphite sequencing
Thermoregulatory pathway underlying the pyrogenic effects of prostaglandin E
2
in the lateral parabrachial nucleus of male rats
期刊论文
ACTA PHARMACOLOGICA SINICA, 2024
作者:
Xu, Jian-hui
;
He, Tian-hui
;
Wang, Nan-ping
;
Gao, Wen-min
;
Cheng, Yong-jing
Adobe PDF(9174Kb)
|
收藏
|
浏览/下载:201/1
|
提交时间:2024/05/14
lateral parabrachial nucleus
preoptic area
fever
PGE(2)
EP3 receptor
A-type potassium current
Efficient Production of 9,22-Dihydroxy-23,24-bisnorchol-4-ene-3-one from Phytosterols by Modifying Multiple Genes in
Mycobacterium fortuitum
期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2024, 卷号: 25, 期号: 7
作者:
Han, Suwan
;
Liu, Xiangcen
;
He, Beiru
;
Zhai, Xinghui
;
Yuan, Chenyang
Adobe PDF(1516Kb)
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收藏
|
浏览/下载:172/0
|
提交时间:2024/05/14
C22 steroids
9,22-dihydroxy-23,24-bisnorchol-4-enehp-3-one(9-OHBA)
Mycobacterium fortuitum
phytosterol
hsd4A
fadA5
KDEL Receptor Trafficking to the Plasma Membrane Is Regulated by ACBD3 and Rab4A-GTP
期刊论文
CELLS, 2023, 卷号: 12, 期号: 7, 页码: 1079
作者:
Tan, Chuanting
;
Du, Yulei
;
Zhu, Lianhui
;
Jing, Shuaiyang
;
Gao, Jingkai
Adobe PDF(40485Kb)
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收藏
|
浏览/下载:363/1
|
提交时间:2023/04/19
KDEL receptor
ACBD3
Rab4A
Rab11A
Golgi
plasma membrane
An A-Kinase Anchoring Protein (ACBD3) Coordinates Traffic-Induced PKA Activation At The Golgi
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2023, 卷号: 299, 期号: 5
作者:
Jia, Jie
;
Tang, Shuocheng
Adobe PDF(23708Kb)
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浏览/下载:335/1
|
提交时间:2023/04/24
Enzymes
A-kinase-anchoring proteins
Acyl-CoA
Acyl-CoA-binding domain-containing 3
Binding domain
Endoplasmic reticulum
Golgi
KDEL receptor
Membrane trafficking
Protein kinase A
Regulatory subunits
Preparation of High-Stability Ceramic Slurry with Gel Behavior for Stereolithography 3D Printing
期刊论文
MATERIALS, 2023, 卷号: 16, 期号: 7
作者:
Wang, Ning
;
Chang, Hai
;
Zhang, Chi
;
Wu, Yingna
;
Yang, Rui
Adobe PDF(4673Kb)
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收藏
|
浏览/下载:3096/1889
|
提交时间:2023/04/28
Elasticity
Gelation
Stability
Stereolithography
3-D printing
3D-printing
A: Ceramics
Ceramic slurry
Gel behavior
Gelling agents
Loss factor
Slurry stability
Stereolithography printing
Three dimensional network structure
Interband transitions of InAs/AlAs Short-Period superlattices grown by molecular beam epitaxy
期刊论文
JOURNAL OF CRYSTAL GROWTH, 2023, 卷号: 605
作者:
Yao, Lu
;
Wang, Wenyang
;
Yao, Jinshan
;
Lu, Kechao
;
Lu, Hong
Adobe PDF(1253Kb)
|
收藏
|
浏览/下载:320/2
|
提交时间:2023/03/10
luminum
Aluminum compounds
III-V semiconductors
Indium
Indium arsenide
Molecular beams
Optical properties
Semiconductor quantum wells
Spectroscopic ellipsometry
A1.
A3.
B1.
B2.
Inter-band transition
Molecular-beam epitaxy
Semiconducting ternary materials
Short period superlattice
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