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Long-range gating regulation by leaflet and autoinhibitory domains in mouse type 1 IP3 receptors 期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2025, 卷号: 766
作者:  Hamada, Kozo;  Terauchi, Akiko
Adobe PDF(2891Kb)  |  收藏  |  浏览/下载:6/1  |  提交时间:2025/05/20
Expanding the utilization of binding pockets proves to be effective for noncovalent small molecule inhibitors against SARS-CoV-2 Mpro 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289
作者:  Yang, Qi;  Huang, Xupeng;  Zhang, Hongbo;  Sun, Jing;  Tang, Jielin
Adobe PDF(5890Kb)  |  收藏  |  浏览/下载:87/9  |  提交时间:2025/04/07
Discovery of novel GluN1/GluN3A NMDA receptor inhibitors using a deep learning-based method 期刊论文
ACTA PHARMACOLOGICA SINICA, 2025
作者:  Wang, Shi-hang;  Zeng, Yue;  Yang, Hao;  Tian, Si-yuan;  Zhou, Yong-qi
Adobe PDF(2216Kb)  |  收藏  |  浏览/下载:10/1  |  提交时间:2025/05/20
Structure and mechanism of a mycobacterial isoniazid efflux pump MsRv1273c/72c with a degenerate nucleotide-binding site 期刊论文
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1
作者:  Yu, Jing;  Lan, Yuhui;  Zhu, Chen;  Chen, Zhendong;  Pan, Junyi
Adobe PDF(5650Kb)  |  收藏  |  浏览/下载:14/1  |  提交时间:2025/05/12
其在制备用于治疗与肠道病毒有关的疾病的化合物以及药物中的用途。 专利
申请号:JP2024559936,申请日期: 2025-04-16,类型:发明申请,状态:实质审查
发明人:  楊海涛;  周浩;  段胤凱;  王鎬鋒;  楊秀娜
Unknown(2120Kb)  |  收藏  |  浏览/下载:38/0  |  提交时间:2025/04/17
Combined treatment targeting Ca2+store mediated Ca2+release and store-operated calcium entry reduces secondary axonal degeneration and improves functional outcome after SCI 期刊论文
EXPERIMENTAL NEUROLOGY, 2025, 卷号: 386
作者:  Jones, Emma;  Ames, Spencer O.;  Brooks, Jesse;  Morehouse, Johnny;  Hill, Norah
Adobe PDF(5086Kb)  |  收藏  |  浏览/下载:94/4  |  提交时间:2025/03/03
高效和特异性的RNA编辑系统 专利
申请号:WOCN24120035,申请日期: 2025-03-27,类型:发明申请,状态:未进入国家阶段-PCT有效期内
发明人:  Chen, Jia;  Yang, Li;  Yang, Bei;  Li, Guangye;  Chen, Guo
收藏  |  浏览/下载:56/0  |  提交时间:2025/03/28
Specific and efficient RNA A-to-I editing through cleavage of an ADAR inhibitor 期刊论文
NATURE BIOTECHNOLOGY, 2025
作者:  Guangye Li;  Guo Chen;  Guo-Hua Yuan;  Jia Wei;  Qingyang Ni
Adobe PDF(11217Kb)  |  收藏  |  浏览/下载:99/7  |  提交时间:2025/03/27
Leveraging base excision repair for efficient adenine base editing of mitochondrial DNA 期刊论文
NATURE BIOTECHNOLOGY, 2025
作者:  Fan, Yuhang;  Xu, Wenchao;  Gao, Bao-Qing;  Qin, Huichao;  Wu, Xiaoyi
Adobe PDF(15428Kb)  |  收藏  |  浏览/下载:46/3  |  提交时间:2025/04/07
化合物及其在制备治疗肠道病毒相关疾病的药物中的应用 专利
申请号:EP23787710,申请日期: 2025-02-19,类型:发明申请,状态:实质审查
发明人:  Yang, Haitao;  Zhou, Hao;  Duan, Yinkai;  Wang, Haofeng
Adobe PDF(922Kb)  |  收藏  |  浏览/下载:80/0  |  提交时间:2025/02/20
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