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Expanding the utilization of binding pockets proves to be effective for noncovalent small molecule inhibitors against SARS-CoV-2 Mpro 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289
作者:  Yang, Qi;  Huang, Xupeng;  Zhang, Hongbo;  Sun, Jing;  Tang, Jielin
Adobe PDF(5890Kb)  |  收藏  |  浏览/下载:79/8  |  提交时间:2025/04/07
Elucidating Contributions of Drug Transporters/Enzyme to Nonlinear Pharmacokinetics of Grazoprevir by PBPK Modeling With a Cluster Gauss-Newton Method 期刊论文
CPT-PHARMACOMETRICS & SYSTEMS PHARMACOLOGY, 2025
作者:  Yoshikado, Takashi;  Aoki, Yasunori;  Nakamura, Ryo;  Shida, Saeko;  Sugiyama, Yuichi
Adobe PDF(1329Kb)  |  收藏  |  浏览/下载:92/3  |  提交时间:2025/02/17
When to consider intra-target microdosing: physiologically based pharmacokinetic modeling approach to quantitatively identify key factors for observing target engagement 期刊论文
FRONTIERS IN PHARMACOLOGY, 2024, 卷号: 15
作者:  Aoki, Yasunori;  Rowland, Malcom;  Sugiyama, Yuichi
Adobe PDF(1837Kb)  |  收藏  |  浏览/下载:374/2  |  提交时间:2024/08/26
Pathway network-based quantitative modeling of the time-dependent and dose-response anti-inflammatory effect of Reduning Injection 期刊论文
JOURNAL OF ETHNOPHARMACOLOGY;, 2023, 卷号: 307
作者:  Xie, Fuda;  Xie, Mingxiang;  Yang, Yibing;  Ao, Weizhen;  Zhao, Tingxiu
Adobe PDF(3150Kb)  |  收藏  |  浏览/下载:388/2  |  提交时间:2023/03/24
Pharmacokinetics and effects of demographic factors on blood 25(OH)D3 levels after a single orally administered high dose of vitamin D3 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 11, 页码: 1509-1515
作者:  Chen, Pei-zhan;  Li, Mian;  Duan, Xiao-hua;  Jia, Jing-ying;  Li, Jing-quan
Adobe PDF(314Kb)  |  收藏  |  浏览/下载:1426/443  |  提交时间:2017/07/04
In silico ADME/T modelling for rational drug design 期刊论文
QUARTERLY REVIEWS OF BIOPHYSICS, 2015, 卷号: 48, 期号: 4, 页码: 488-515
作者:  Wang, Yulan;  Xing, Jing;  Xu, Yuan;  Zhou, Nannan;  Peng, Jianlong
Adobe PDF(829Kb)  |  收藏  |  浏览/下载:475/0  |  提交时间:2017/07/04
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