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Discovery of novel and highly potent anticancer agents enabled by selenium scanning of noscapine
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 293
作者:
Li, Defeng
;
Shen, Shuting
;
Liu, Chuanxu
;
Guo, Tingyu
;
Liu, Yuhuan
Adobe PDF(19864Kb)
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浏览/下载:41/8
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提交时间:2025/05/26
Noscapine
Selenium scanning
Anticancer activity
p53
DNA damage response
Mitochondrial dysfunction
Manifold-valued models for analysis of EEG time series data
期刊论文
COMPUTATIONAL STATISTICS AND DATA ANALYSIS, 2025, 卷号: 209
作者:
Ding, Tao
;
Nye, Tom M.W.
;
Wang, Yujiang
Adobe PDF(4588Kb)
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浏览/下载:67/1
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提交时间:2025/04/11
Electrocardiography
Gaussian noise (electronic)
Matrix algebra
Maximum likelihood estimation
Time series
Time series analysis
Vector spaces
Auto-regressive
Brain electrical activity
Clinical tools
Covariance matrices
Mean-reversion
Modeling results
Neuroscience
Riemannian manifold
Time-series data
Times series
Systematic trans-Activity Comparison of Several Reported Cas12f Nucleases
期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2025, 卷号: 43, 期号: 12, 页码: 1339-1347
作者:
Wang YN(王艳男)
;
Tang N(汤娜)
;
Ji QJ(季泉江)
Adobe PDF(2363Kb)
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浏览/下载:79/8
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提交时间:2025/03/31
Cas12f
Trans-cleavage activity
cis-Cleavage activity
In vitro diagnostics
In vivo genome editing
Discovery and biological evaluation of carborane-containing derivatives as TEAD auto palmitoylation inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 121
作者:
Li, Chaofan
;
Zhang, Yingshuang
;
Zhang, Ziyin
;
Zhang, Yirong
;
Song, Yuxuan
Adobe PDF(3973Kb)
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浏览/下载:102/7
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提交时间:2025/03/18
TEAD
Palmitoylation inhibitor
Carborane
Anti-cancer activity
Computationally revisiting pH- and ligand-dependence of Fenton reaction selectivity and activity in aqueous solution
期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2025
作者:
Liu, Ying
;
Hu, Peijun
;
Wang, Haifeng
Adobe PDF(2463Kb)
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浏览/下载:12/0
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提交时间:2025/06/17
Binding sites
Degradation
Deprotonation
Free radical reactions
Oxidation
Reaction intermediates
Reaction kinetics
Atomic levels
Bond cleavages
Catalyse
Fe complexes
Fe-based
Fenton reactions
PH-dependent
Reaction activity
Reaction selectivity
Reactive oxidative species
Enzyme Surface Residues Direct Encapsulation into Metal–Organic Frameworks for Performance Regulation
期刊论文
ANGEWANDTE CHEMIE - INTERNATIONAL EDITION, 2025, 卷号: 64, 期号: 20
作者:
Wu, Mengyao
;
Du, Yuexin
;
Xu, Hui
;
Zhang, Xiehaoran
;
Ma, Jialong
Adobe PDF(11670Kb)
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浏览/下载:94/4
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提交时间:2025/03/14
Crystalline materials - Enzyme activity - Enzyme immobilization - Metal-Organic Frameworks
Cytochrome c - Enzyme catalysis - Immobilisation - Metalorganic frameworks (MOFs) - Modified proteins - Performance - Structure-activity relationships - Surface residues - Surface-modification - Template synthesis
metal-organic frameworks
enzyme catalysis
template synthesis
immobilization
structure-activity relationships
Conformational restriction enables discovering a series of chroman derivatives as potent and selective Nav1.8 inhibitors with improved pharmacokinetic properties
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 293, 页码: 117697
作者:
Li, Na
;
Wang, Linlin
;
Hu, Xinyuan
;
Xu, Haiyan
;
Yang, Bowen
Adobe PDF(4737Kb)
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浏览/下载:22/4
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提交时间:2025/05/20
Voltage-gated sodium channel 1.8
Conformational restriction
Pharmacokinetic
Structure-activity relationship
Analgesic
Expanding the utilization of binding pockets proves to be effective for noncovalent small molecule inhibitors against SARS-CoV-2 Mpro
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289
作者:
Yang, Qi
;
Huang, Xupeng
;
Zhang, Hongbo
;
Sun, Jing
;
Tang, Jielin
Adobe PDF(5890Kb)
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浏览/下载:105/10
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提交时间:2025/04/07
SARS-CoV-2
M pro inhibitors
Pharmacokinetics properties
In vivo antiviral activity
Structure-activity relationship analysis of meta-substituted N-cyclopropylmethyl-nornepenthones with mixed KOR/MOR activities
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289
作者:
Tang, Siyuan
;
Hu, Shuyang
;
Feng, Lijing
;
Kong, Linghui
;
Gui, Jiangwen
Adobe PDF(2887Kb)
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收藏
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浏览/下载:57/1
|
提交时间:2025/03/25
N-Cyclopropylmethyl-nornepenthones
Structure-activity relationship
MOR antagonist
KOR agonist
Substance use disorder
Rapid and In Situ Active Sites Regeneration for OER Activity Recovery and Greatly Prolonged Water-Splitting Performance
期刊论文
ANGEWANDTE CHEMIE - INTERNATIONAL EDITION, 2025, 卷号: 64, 期号: 21
作者:
Li, Qin
;
Luo, Wenshu
;
Cui, Xiangzhi
;
Shi, Jianlin
Adobe PDF(5729Kb)
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收藏
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浏览/下载:19/2
|
提交时间:2025/04/25
Abiotic
Anthropogenic
Electrochemical oxidation
Electrolytic cells
Nickel
Nickel coatings
Redox reactions
Active site
Active site regeneration
Activity recovery
Evolution reactions
Initial activity
Nickel mesh
Oxygen evolution
Reaction activity
Water splitting
]+ catalyst
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