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Discovery of novel GluN1/GluN3A NMDA receptor inhibitors using a deep learning-based method
期刊论文
ACTA PHARMACOLOGICA SINICA, 2025
作者:
Wang, Shi-hang
;
Zeng, Yue
;
Yang, Hao
;
Tian, Si-yuan
;
Zhou, Yong-qi
Adobe PDF(2216Kb)
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收藏
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浏览/下载:18/2
|
提交时间:2025/05/20
N
-methyl-
D
-aspartate receptors
GluN1/GluN3A
ligand-based virtual screening
scaffold hopping
deep learning
GeminiMol
Fine-tuning phenoxy silyl scaffolds for the development of glutathione-responsive prodrugs and antibody-drug conjugates
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 120
作者:
Wei, Ding
;
Wang, Huihui
;
Huangfu, Shangwei
;
Qi, Cheng
;
Jiang, Yuecheng
Adobe PDF(5369Kb)
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浏览/下载:100/7
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提交时间:2025/03/03
Phenoxy silyl scaffold
Antibody-drug conjugate
Prodrug
GSH-cleavage
VitisC: Visualizing interested target via integrated scaffold of cytoophidium
预印本
2025
作者:
Yin, Boqi
;
Hu, Huan-Huan
;
Zhong, Jiale
;
Liu, Ji-Long
收藏
|
浏览/下载:56/0
|
提交时间:2025/03/25
cryo-EM
CTP synthase
cytoophidium
the scaffold of cytoophidium
VitisC
Design and synthesis of Thieno[3, 2-b]pyridinone derivatives exhibiting potent activities against
Mycobacterium tuberculosis
in vivo by targeting Enoyl-ACP reductase
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 279
作者:
Liang, Lihong
;
Liu, Zhiyong
;
Chen, Jie
;
Zha, Qin
;
Zhou, Yihuan
Adobe PDF(1929Kb)
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浏览/下载:316/3
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提交时间:2024/09/30
Thieno[3, 2-b]pyridinone
Anti-Tuberculosis activity
Scaffold hopping
InhA
InhA
Discovery of Novel BCL6-Targeting PROTACs with Effective Antitumor Activities against DLBCL in Vitro and in Vivo
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 277
作者:
Dazhao Mi
;
Cheng Li(李成)
;
Yuzhan Li
;
Mingyue Yao
;
Yan Li
Adobe PDF(7740Kb)
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浏览/下载:393/13
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提交时间:2024/09/02
BCL6
PROTACs
DLBCL
Pyrimidinamine scaffold
Lead compound
Spatiotemporal Regulation of Injectable Heterogeneous Silk Gel Scaffolds for Accelerating Guided Vertebral Repair
期刊论文
ADVANCED HEALTHCARE MATERIALS, 2023, 卷号: 12, 期号: 7
作者:
Wang, Tianji
;
Liu, Keyin
;
Wang, Jing
;
Xiang, Geng
;
Hu, Xiaofan
Adobe PDF(2994Kb)
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浏览/下载:270/0
|
提交时间:2023/02/24
angiogenesis
bone regeneration
HIF-1 alpha stabilization
injectable heterogeneous silk gel scaffold
spatiotemporal sustained drug release
vertebral augmentation
In Situ Regulation of Macrophage Polarization to Enhance Osseointegration Under Diabetic Conditions Using Injectable Silk/Sitagliptin Gel Scaffolds
期刊论文
ADVANCED SCIENCE, 2021
作者:
Xiang, Geng
;
Liu, Keyin
;
Wang, Tianji
;
Hu, Xiaofan
;
Wang, Jing
Adobe PDF(4969Kb)
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浏览/下载:519/0
|
提交时间:2021/01/19
diabetes mellitus
injectable silk gel scaffold
macrophage polarization
osseointegration promotion
3D Silk-Based Bioelectronic Scaffolds for Osteochondral Regeneration
会议论文
33RD IEEE INTERNATIONAL CONFERENCE ON MICRO ELECTRO MECHANICAL SYSTEMS, MEMS 2020, Vancouver, BC, Canada, JAN 18-22, 2020
作者:
Gao, Zhiheng
;
Li, Shengkun
;
Chen, Fang
;
Hua, Yinghui
;
Tao, Tiger H.
Adobe PDF(1160Kb)
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浏览/下载:704/4
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提交时间:2020/06/17
Silk Scaffold
Multi-layer Structure
Osteochondral Regeneration
Photocrosslinked hydrogels from coumarin derivatives of hyaluronic acid for tissue engineering applications
期刊论文
MATERIALS SCIENCE & ENGINEERING C-MATERIALS FOR BIOLOGICAL APPLICATIONS, 2019, 卷号: 96, 页码: 625-634
作者:
Beninatto, Riccardo
;
Barbera, Carlo
;
De Lucchi, Ottorino
;
Borsato, Giuseppe
;
Serena, Elena
Adobe PDF(2063Kb)
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浏览/下载:542/3
|
提交时间:2018/12/17
Hyaluronic acid
Hydrogel
Scaffold
Coumarin
Photocrosslinking
Tissue engineering
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