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期刊影响因子降序
Synthesis and Biological Evaluation of β‐Lactam Derivatives Targeting Speckle-Type POZ Protein (SPOP)
期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2024
作者:
Chenmao Zhou
;
Xinyue Hao
;
Zhengyang Chen
;
Runze Zhang
;
Qian Zhou
Adobe PDF(3478Kb)
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收藏
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浏览/下载:140/0
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提交时间:2024/11/27
Speckle-type POZ protein (SPOP)
SPOP inhibitors
Clear cell renal cell carcinoma (ccRCC)
Structure−activity relationship (SAR)
Structure and biochemical characterization of L-2-hydroxyglutarate dehydrogenase and its role in the pathogenesis of L-2-hydroxyglutaric aciduria
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2024, 卷号: 300, 期号: 1
作者:
Yang, Jun
;
Chen, Xingchen
;
Jin, Shan
;
Ding, Jianping
Adobe PDF(3335Kb)
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收藏
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浏览/下载:384/0
|
提交时间:2024/01/19
Catalyst activity
Mitochondria
2-hydroxyglutaric aciduria
2-oxoglutarate
Biochemical characterization
Catalytic mechanisms
Drosophilla melanogaster
L-2-hydroxyglutarate dehydrogenase
Mitochondrial membranes
Protein crystallography
Structure characterization
Substrate specificity
Affinity-based protein profiling-driven discovery of myricanol as a Nampt activator
期刊论文
BIOORGANIC CHEMISTRY;, 2023, 卷号: 133
作者:
Lyu, Peng
;
Li, Shengrong
;
Han, Ying
;
Shen, Shengnan
;
Feng, Zheling
Adobe PDF(3298Kb)
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浏览/下载:322/0
|
提交时间:2023/03/24
Activity-based protein profiling
Myotubes
Myricanol
Nampt
Photo-affinity probe
Cell-Free Expression of a Therapeutic Protein Serratiopeptidase
期刊论文
MOLECULES, 2023, 卷号: 28, 期号: 7, 页码: 3132
作者:
Meng, Yaru
;
Yang, Miaomiao
;
Liu, Wanqiu
;
Li, Jian
Adobe PDF(1924Kb)
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浏览/下载:507/0
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提交时间:2023/05/09
cell-free protein synthesis
therapeutic proteins
serratiopeptidase
enzymatic activity
cell-free synthetic biology
Molecular mechanism of S-adenosylmethionine sensing by SAMTOR in mTORC1 signaling
期刊论文
SCIENCE ADVANCES, 2022, 卷号: 8, 期号: 26
作者:
Tang, Xin
;
Zhang, Yifan
Adobe PDF(3660Kb)
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浏览/下载:646/8
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提交时间:2022/07/25
Amino-acids
Binding-sites
GTPase-activating protein
Helical domains
Mechanistics
Methyltransferases
Molecular mechanism
Protein activity
S-adenosylmethionine
Target of rapamycin
Ligand-Directed Caging Enables the Control of Endogenous DNA Alkyltransferase Activity with Light inside Live Cells
期刊论文
ANGEWANDTE CHEMIE - INTERNATIONAL EDITION, 2022, 卷号: 61, 期号: 17
作者:
Zhang, Yixin
;
Han, Lili
;
Tian, Xiaoxu
;
Peng, Chao
;
Chen, Yiyun
Adobe PDF(3076Kb)
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浏览/下载:644/0
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提交时间:2022/03/18
Amino acids
Cytology
DNA
Irradiation
Ligands
Mammals
Modulation
Alkyltransferase
DNA alkyltransferase
Endogenous protein modulation
Light irradiations
Live cell
Molecule ligands
Photodecaging
Protein activity
Small molecules
Small-molecule-ligand
Modulating effects of RAMPs on signaling profiles of the glucagon receptor family
期刊论文
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 2
作者:
Shao, Lijun
;
Chen, Yan
;
Zhang, Shikai
;
Zhang, Zhihui
;
Cao, Yongbing
Adobe PDF(3846Kb)
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浏览/下载:402/1
|
提交时间:2022/03/23
G protein-coupled receptor
Glucagon receptor family
Receptor activity-modulating protein
Signaling
Allosteric modulation
GPCR-RAMP interaction
Receptor pharmacology
Ligand selectivity
Designing Modular Cell-free Systems for Tunable Biotransformation of L-phenylalanine to Aromatic Compounds
期刊论文
FRONTIERS IN BIOENGINEERING AND BIOTECHNOLOGY, 2021, 卷号: 9
作者:
Yang, Chen
;
Liu, Yushi
;
Liu, Wan-Qiu
;
Wu, Changzhu
;
Li, Jian
Adobe PDF(1836Kb)
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收藏
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浏览/下载:831/290
|
提交时间:2021/08/20
cell-free systems
biocatalysis
biotransformation
value-added chemicals
synthetic biology
Amino acids
Aromatic compounds
Biochemistry
Bioconversion
Biosynthesis
Catalyst activity
Cells
Enzymes
Escherichia coli
Biosynthetic pathway
Cell free protein synthesis
Cell
free reactions
free system
Conversion rates
Enzymatic pathways
Resource limitations
Value
added chemicals
Allosteric inhibition of CRISPR-Cas9 by bacteriophage-derived peptides
期刊论文
GENOME BIOLOGY, 2020, 卷号: 21, 期号: 1
作者:
Cui, Yan-ru
;
Wang, Shao-jie
;
Chen, Jun
;
Li, Jie
;
Chen, Wenzhang
Adobe PDF(2515Kb)
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收藏
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浏览/下载:657/1
|
提交时间:2020/03/28
CRISPR-Cas9
Inoviridae bacteriophage
Major coat protein G8P
Allosteric inhibition
Off-target activity
Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 163, 页码: 281-294
作者:
Xing, Jing
;
Zhang, Rukang
;
Jiang, Xiangrui
;
Hu, Tianwen
;
Wang, Xinjun
Adobe PDF(4202Kb)
|
收藏
|
浏览/下载:459/1
|
提交时间:2019/03/04
Bromodomain-containing protein 4
8-OH-Quinoline
Anti-cancer activity
Rational hit-to-lead optimization
Computer-aided drug design
Early ADME/T evaluation
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