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IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response 期刊论文
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2025, 卷号: 14, 期号: 1
作者:  Yao, Mingyue;  Yan, Wenzhong;  Wang, Yafang;  Zhao, Yu;  Xu, Xiaowei
Adobe PDF(14589Kb)  |  收藏  |  浏览/下载:82/3  |  提交时间:2025/03/03
Targeted Degradation of SOS1 Exhibits Potent Anticancer Activity and Overcomes Resistance in KRAS-Mutant Tumors and BCR-ABL-Positive Leukemia 期刊论文
CANCER RESEARCH, 2025, 卷号: 85, 期号: 1
作者:  Luo, Ziwei;  Lin, Chencen;  Yu, Chuwei;  Yuan, Changxian;  Wu, Wenyong
Adobe PDF(22554Kb)  |  收藏  |  浏览/下载:170/4  |  提交时间:2025/01/13
Mutation in CDC42 Gene Set as a Response Biomarker for Immune Checkpoint Inhibitor Therapy 期刊论文
CANCER MEDICINE, 2025, 卷号: 14, 期号: 1
作者:  Wang, Kun;  Zhang, Yingying;  Su, Zhaoming;  Wang, Bei;  Zhou, Yuanyang
Adobe PDF(6595Kb)  |  收藏  |  浏览/下载:125/1  |  提交时间:2025/01/20
Concurrent inhibition of p300/CBP and FLT3 enhances cytotoxicity and overcomes resistance in acute myeloid leukemia 期刊论文
ACTA PHARMACOLOGICA SINICA, 2025
作者:  Chen, Yu-jun;  Zhao, Yu;  Yao, Ming-yue;  Wang, Ya-fang;  Ma, Ming
Adobe PDF(6202Kb)  |  收藏  |  浏览/下载:95/7  |  提交时间:2025/02/12
SOS1蛋白降解剂及其应用 专利
申请号:CN202310427933.8,申请日期: 2024-10-22,类型:发明申请,状态:实质审查
发明人:  谢成英;  姜标;  杨小宝
Adobe PDF(5367Kb)  |  收藏  |  浏览/下载:348/0  |  提交时间:2024/10/22
Discovery of Novel BCL6-Targeting PROTACs with Effective Antitumor Activities against DLBCL in Vitro and in Vivo 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 277
作者:  Dazhao Mi;  Cheng Li(李成);  Yuzhan Li;  Mingyue Yao;  Yan Li
Adobe PDF(7740Kb)  |  收藏  |  浏览/下载:364/13  |  提交时间:2024/09/02
五环三萜衍生物的医药用途、五环三萜衍生物、包含其的药物组合物 专利
申请号:CN202311207625.0,申请日期: 2024-03-22,类型:发明申请,状态:公开
发明人:  梅良和;  谢成英;  白芳;  王亚芳;  徐岚松
Adobe PDF(8828Kb)  |  收藏  |  浏览/下载:500/1  |  提交时间:2024/03/22
Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers 期刊论文
ADVANCED SCIENCE, 2024, 卷号: 11, 期号: 41
作者:  Wang, Yafang;  Xu, Lansong;  Ling, Lijun;  Yao, Mingyue;  Shi, Shangxuan
Adobe PDF(9804Kb)  |  收藏  |  浏览/下载:351/2  |  提交时间:2024/09/20
Targeting ST8SIA6-AS1 counteracts KRASG12C inhibitor resistance through abolishing the reciprocal activation of PLK1/c-Myc signaling 期刊论文
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2023
作者:  Yafang Wang;  Mingyue Yao;  Cheng Li (李成);  Kexin Yang;  Xiaolong Qin
Adobe PDF(16153Kb)  |  收藏  |  浏览/下载:378/5  |  提交时间:2024/09/02
Mechanism of hormone and allosteric agonist mediated activation of follicle stimulating hormone receptor 期刊论文
NATURE COMMUNICATIONS;, 2023, 卷号: 14, 期号: 1
作者:  Duan, Jia
Adobe PDF(3025Kb)  |  收藏  |  浏览/下载:1085/188  |  提交时间:2023/03/24
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