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Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening 期刊论文
RSC ADVANCES, 2019, 卷号: 9, 期号: 9, 页码: 4917-4924
Authors:  Tao, Hongru;  Wang, Jun;  Lu, Wenchao;  Zhang, Rukang;  Xie, Yiqian;  Liu, Yu-Chih;  Liu, Rongfeng;  Yue, Liyan;  Chen, Kaixian;  Jiang, Hualiang;  Zhang, Yuanyuan;  Xu, Xiaohui;  Luo, Cheng
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Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues 期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2017, 卷号: 15, 期号: 44, 页码: 9352-9361
Authors:  Jiang, Hao;  Xing, Jing;  Wang, Chen;  Zhang, Hao;  Yue, Liyan;  Wan, Xiaozhe;  Chen, Wei;  Ding, Hong;  Xie, Yiqian;  Tao, Hongru;  Chen, Zhifeng;  Jiang, Hualiang;  Chen, Kaixian;  Chen, Shijie;  Zheng, Mingyue;  Zhang, Yuanyuan;  Luo, Cheng
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Development of Potent Type I Protein Arginine Methyltransferase (PRMT) Inhibitors of Leukemia Cell Proliferation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 21, 页码: 8888-8905
Authors:  Wang, Chen;  Jiang, Hao;  Jin, Jia;  Xie, Yiqian;  Chen, Zhifeng;  Zhang, Hao;  Lian, Fulin;  Liu, Yu-Chih;  Zhang, Chenhua;  Ding, Hong;  Chen, Shijie;  Zhang, Naixia;  Zhang, Yuanyuan;  Jiang, Hualiang;  Chen, Kaixian;  Ye, Fei;  Yao, Zhiyi;  Luo, Cheng
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Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay 期刊论文
MEDCHEMCOMM, 2017, 卷号: 8, 期号: 6, 页码: 1322-1331
Authors:  Chen, Zhifeng;  Zhang, Hao;  Liu, Shien;  Xie, Yiqian;  Jiang, Hao;  Lu, Wenchao;  Xu, Heng;  Yue, Liyan;  Zhang, Yuanyuan;  Ding, Hong;  Zheng, Mingyue;  Yu, Kunqian;  Chen, Kaixian;  Jiang, Hualiang;  Luo, Cheng
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Discovery of novel BRD4 inhibitors by high-throughput screening, crystallography, and cell-based assays 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 9, 页码: 2003-2009
Authors:  Sun, Zhongya;  Zhang, Hao;  Chen, Zhifeng;  Xie, Yiqian;  Jiang, Hao;  Chen, Limin;  Ding, Hong;  Zhang, Yuanyuan;  Jiang, Hualiang;  Zheng, Mingyue;  Luo, Cheng
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Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 20, 页码: 8166-8181
Authors:  Meng, Fanwang;  Cheng, Sufang;  Ding, Hong;  Liu, Shien;  Liu, Yan;  Zhu, Kongkai;  Chen, Shijie;  Lu, Junyan;  Xie, Yiqian;  Li, Linjuan;  Liu, Rongfeng;  Shi, Zhe;  Zhou, Yu;  Liu, Yu-Chih;  Zheng, Mingyue;  Jiang, Hualiang;  Lu, Wencong;  Liu, Hong;  Luo, Cheng
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