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Access to N-Alkylazaheterocyclic Salts by Activation of Alkoxy C-O Bonds in Polyol Esters 期刊论文
THE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 88, 期号: 14, 页码: 9769-9782
作者:  Shi, Zhan;  Bian, Qiang;  Li, Zhi
Adobe PDF(3266Kb)  |  收藏  |  浏览/下载:564/0  |  提交时间:2023/07/10
Design and synthesis of novel benzimidazole-iminosugars linked a substituted phenyl group and their inhibitory activities against beta-glucosidase 期刊论文
BIOORGANIC CHEMISTRY, 2022, 卷号: 127
作者:  Liu, Xu;  Li, Fengxin;  Su, Lulu;  Wang, Mingchen;  Jia, Tongguan
Adobe PDF(2594Kb)  |  收藏  |  浏览/下载:354/0  |  提交时间:2022/08/15
Hypervalent Iodine Reagents Enable C(sp(2))-H Amidation of (Hetero)arenes with Iminophenylacetic Acids 期刊论文
ORGANIC LETTERS, 2022
作者:  Pan, Yue;  Liu, Zhengyi;  Zou, Peng;  Chen, Yali;  Chen, Yiyun
Adobe PDF(1799Kb)  |  收藏  |  浏览/下载:552/0  |  提交时间:2022/09/19
Selenylation Chemistry Suitable for On-Plate Parallel and On-DNA Library Synthesis Enabling High-Throughput Medicinal Chemistry 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022
作者:  Xu, Hongtao;  Wang, Yan;  Dong, Hewei;  Zhang, Yiyuan;  Gu, Yuang
Adobe PDF(11674Kb)  |  收藏  |  浏览/下载:773/6  |  提交时间:2022/07/01
Discovery of Small-Molecule Degraders of the CDK9-Cyclin T1 Complex for Targeting Transcriptional Addiction in Prostate Cancer 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2022
作者:  Li, Jiacheng;  Liu, Ting;  Song, Yuanli;  Wang, Mingyu;  Liu, Liping
Adobe PDF(11347Kb)  |  收藏  |  浏览/下载:425/1  |  提交时间:2022/08/23
Hypervalent Iodine Reagents Enable C-H Alkynylation with Iminophenylacetic Acids via Alkoxyl Radicals 期刊论文
ORGANIC LETTERS, 2022, 卷号: 24, 期号: 32
作者:  Liu, Zhengyi;  Pan, Yue;  Zou, Peng;  Huang, Hanchu;  Chen, Yali
Adobe PDF(1753Kb)  |  收藏  |  浏览/下载:572/0  |  提交时间:2022/09/05
Reactive oxygen species-responsive Pre-PROTAC for tumor-specific protein degradation 期刊论文
CHEMICAL COMMUNICATIONS, 2022, 卷号: 58, 期号: 72, 页码: 10072-10075
作者:  Liu, Haixia;  Ren, Chaowei;  Sun, Renhong;  Wang, Huihui;  Zhan, Yuexiong
Adobe PDF(967Kb)  |  收藏  |  浏览/下载:666/7  |  提交时间:2022/08/29
Visible-light-promoted S-trifluoromethylation of thiophenols with trifluoromethyl phenyl sulfone 期刊论文
CHEMICAL COMMUNICATIONS, 2022
作者:  Wei, Zhiqiang;  Lou, Zhengzhao;  Ni, Chuanfa;  Zhang, Wei;  Hu, Jinbo
Adobe PDF(1038Kb)  |  收藏  |  浏览/下载:409/1  |  提交时间:2022/08/29
Design, synthesis and biological evaluation of novel osimertinib derivatives as reversible EGFR kinase inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 238
作者:  Ding, Shi;  Gao, Ziye;  Hu, Ziqiang;  Qi, Rui;  Zheng, Xiangshan
Adobe PDF(8843Kb)  |  收藏  |  浏览/下载:384/0  |  提交时间:2022/08/15
Iridium-Catalyzed Selective trans-Semihydrogenation of 1,3-Enynes with Ethanol: Access to (E,E)-1,4-Diarylbutadienes 期刊论文
ORGANIC LETTERS, 2022, 卷号: 24, 期号: 29
作者:  Huang, Fengjie;  Huang, Zhidao;  Liu, Guixia;  Huang, Zheng
Adobe PDF(1678Kb)  |  收藏  |  浏览/下载:330/0  |  提交时间:2022/08/15
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