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浏览/检索结果: 共23条,第1-10条 帮助

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Discovery of Novel BCL6-Targeting PROTACs with Effective Antitumor Activities against DLBCL in Vitro and in Vivo 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 277
作者:  Dazhao Mi;  Cheng Li(李成);  Yuzhan Li;  Mingyue Yao;  Yan Li
Adobe PDF(7740Kb)  |  收藏  |  浏览/下载:409/13  |  提交时间:2024/09/02
超薄超导NbSe2的点接触安德列夫反射谱研究 学位论文
上海: 上海科技大学, 2021
作者:  雷陇彪
Adobe PDF(2953Kb)  |  收藏  |  浏览/下载:118/0  |  提交时间:2021/11/13
Activation of unfolded protein response overcomes Ibrutinib resistance in diffuse large B-cell lymphoma 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021
作者:  Zhang, Xiao-tuan;  Hu, Xiao-bei;  Wang, Han-lin;  Kan, Wei-juan;  Xu, Lei
Adobe PDF(2353Kb)  |  收藏  |  浏览/下载:325/0  |  提交时间:2020/09/18
The transport properties of ultrathin 2H–NbSe2 期刊论文
SUPERCONDUCTOR SCIENCE & TECHNOLOGY, 2021, 卷号: 24, 期号: 2, 页码: #VALUE!
作者:  L B Lei;  C Zhang;  A B Yu;  W Peng;  H Xiao
Adobe PDF(837Kb)  |  收藏  |  浏览/下载:616/3  |  提交时间:2021/04/29
Design and synthesis of Imidazo[1,2-b]pyridazine IRAK4 inhibitors for the treatment of mutant MYD88 L265P diffuse large B-cell lymphoma 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 190
作者:  Chen, Yun;  Bai, Gang;  Ning, Yi;  Cai, Shi;  Zhang, Tao
Adobe PDF(1964Kb)  |  收藏  |  浏览/下载:342/0  |  提交时间:2020/04/12
Discovery and biological evaluation of N-(3-(7-((2-methoxy-4-(4-methylpiperazin-1-yl)phenyl)amino)-4-methyl-2-oxo-2H-pyrimido[4,5-d][1,3]oxazin-1(4H)-yl)phenyl)acrylamide as potent Bruton's tyrosine kinase inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 415-422
作者:  Lai, Meng-zhen;  Song, Pei-ran;  Dou, Dou;  Diao, Yan-yan;  Tong, Lin-jiang
Adobe PDF(3317Kb)  |  收藏  |  浏览/下载:427/0  |  提交时间:2020/03/16
Discovery and Development of a Series of Pyrazolo[3,4-d]pyridazinone Compounds as the Novel Covalent Fibroblast Growth Factor Receptor Inhibitors by the Rational Drug Design 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 16, 页码: 7473-7488
作者:  Wang, Yulan;  Dai, Yang;  Wu, Xiaowei;  Li, Fei;  Liu, Bo
Adobe PDF(3590Kb)  |  收藏  |  浏览/下载:670/14  |  提交时间:2019/09/10
Discovery and Biological evaluation of pyrimido[4,5-d] pyrimidine-2,4(1H, 3H)-dione derivatives as potent Bruton's tyrosine kinase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3390-3395
作者:  Diao, Yanyan;  Fang, Xiaoyu;  Song, Peiran;  Lai, Mengzhen;  Tong, Linjiang
Adobe PDF(2955Kb)  |  收藏  |  浏览/下载:502/9  |  提交时间:2019/08/20
Chemoselective Synthesis of Lenalidomide-Based PROTAC Library Using Alkylation Reaction 期刊论文
ORGANIC LETTERS, 2019, 卷号: 21, 期号: 10, 页码: 3838-3841
作者:  Qiu, Xing;  Sun, Ning;  Kong, Ying;  Li, Yan;  Yang, Xiaobao
Adobe PDF(1579Kb)  |  收藏  |  浏览/下载:944/21  |  提交时间:2019/06/06
Optimization of novel benzofuro[3,2-b]pyridin-2(1H)-one derivatives as dual inhibitors of BTK and PI3K delta 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 304-316
作者:  Liu, Linyi;  Li, Xinyu;  Cheng, Yu;  Wang, Lianjian;  Yang, Huizhu
Adobe PDF(2749Kb)  |  收藏  |  浏览/下载:563/2  |  提交时间:2019/02/25
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