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Structure-activity relationship analysis of meta-substituted N-cyclopropylmethyl-nornepenthones with mixed KOR/MOR activities
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289
作者:
Tang, Siyuan
;
Hu, Shuyang
;
Feng, Lijing
;
Kong, Linghui
;
Gui, Jiangwen
Adobe PDF(2887Kb)
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浏览/下载:45/1
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提交时间:2025/03/25
N-Cyclopropylmethyl-nornepenthones
Structure-activity relationship
MOR antagonist
KOR agonist
Substance use disorder
Discovery of novel covalent stabilizers for p53 Y220C using structure-based drug discovery methods
期刊论文
MOLECULAR DIVERSITY, 2025
作者:
Wen, Yiming
;
Xu, Peijia
;
Chen, Yijie
;
Meng, Jingyi
;
Zheng, Mingyue
Adobe PDF(4175Kb)
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浏览/下载:75/2
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提交时间:2025/03/03
p53 Y220C
Covalent stabilizer
Virtual screening
Molecular dynamics
DNA binding
Structure-activity relationship
Cancer therapy
Design, Synthesis and Biological Activity Study of γ-Aminobutyric Acid (GABA) Derivatives Containing Bridged Bicyclic Skeletons as BCAT1 Inhibitors
期刊论文
MOLECULES, 2025, 卷号: 30, 期号: 4
作者:
Adobe PDF(2448Kb)
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浏览/下载:57/1
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提交时间:2025/03/10
BCAT1 inhibitor
structure-activity relationship
cancer resistance
third-generation EGFR TKI
GABA
amino acid
bicyclo[3.2.1]octane
Enzyme Surface Residues Direct Encapsulation into Metal–Organic Frameworks for Performance Regulation
期刊论文
ANGEWANDTE CHEMIE - INTERNATIONAL EDITION, 2025
作者:
Wu, Mengyao
;
Du, Yuexin
;
Xu, Hui
;
Zhang, Xiehaoran
;
Ma, Jialong
Adobe PDF(11670Kb)
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浏览/下载:76/3
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提交时间:2025/03/14
Crystalline materials - Enzyme activity - Enzyme immobilization - Metal-Organic Frameworks
Cytochrome c - Enzyme catalysis - Immobilisation - Metalorganic frameworks (MOFs) - Modified proteins - Performance - Structure-activity relationships - Surface residues - Surface-modification - Template synthesis
metal-organic frameworks
enzyme catalysis
template synthesis
immobilization
structure-activity relationships
Inhibitor Development for α‑Synuclein Fibril's Disordered Region to Alleviate Parkinson's Disease Pathology
期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 卷号: 146, 期号: 41, 页码: 28282-28295
作者:
Zhang, Shenqing
;
Xiang, Huaijiang
;
Tao, Youqi
;
Li, Juan
;
Zeng, Shuyi
Adobe PDF(12245Kb)
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浏览/下载:383/14
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提交时间:2024/09/27
Neurodegenerative diseases
Nuclear magnetic resonance spectroscopy
Targeted drug delivery
Amyloid fibril
Disordered regions
EM techniques
High throughput screening
Intrinsically disordered regions
Membrane receptors
Pathological effects
Solid state NMR
Structure-activity relationships
α-synuclein
Cu-OFF/ERI Zeolite: Intergrowth Structure Synergistically Boosting Selective Catalytic Reduction of NOx with NH3
期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2024, 卷号: 146, 期号: 11, 页码: 7605-7615
作者:
Han, Jinfeng
;
Li, Junyan
;
Zhao, Wenru
;
Li, Lin
;
Chen, Mengyang
Adobe PDF(7346Kb)
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浏览/下载:253/1
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提交时间:2024/04/12
Ammonia
Catalyst activity
Copper compounds
Density functional theory
Nitrogen oxides
Selective catalytic reduction
Temperature
Cu based zeolites
Density-functional theory calculations
Diesel exhausts
Intergrowth
Intergrowth structure
NO x
Offretite
Organic templates
Organotemplate-free
Selective catalytic reduction of NO
Synthesis and Biological Evaluation of β‐Lactam Derivatives Targeting Speckle-Type POZ Protein (SPOP)
期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2024
作者:
Chenmao Zhou
;
Xinyue Hao
;
Zhengyang Chen
Adobe PDF(3478Kb)
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浏览/下载:142/0
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提交时间:2024/11/27
Speckle-type POZ protein (SPOP)
SPOP inhibitors
Clear cell renal cell carcinoma (ccRCC)
Structure−activity relationship (SAR)
Strong Metal-Support Interactions: From Characterization, Manipulation to Application in Fischer-Tropsch Synthesis and Atmospheric CO2 hydrogenation
期刊论文
CHEMCATCHEM, 2024, 卷号: 16, 期号: 15
作者:
Zhang, Wenzhe
;
Lin, Heyun
;
An, Yunlei
;
Lin, Tiejun
;
Zhong, Liangshu
Adobe PDF(5691Kb)
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收藏
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浏览/下载:279/1
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提交时间:2024/02/23
Carbon dioxide
Chemical shift
Fischer-Tropsch synthesis
Metal nanoparticles
Water gas shift
Atmospheric CO 2
Characterization techniques
COx hydrogenation
Interaction effect
Interaction phenomena
Metal-support interactions
Overlayers
Strong metal-support interaction
Structural sensitivity
Structure-activity relationships
Mechanism and structure-activity relationship of H2 and CO2 activation at the ZnO/Cu catalyst interface
期刊论文
CATALYSIS SCIENCE AND TECHNOLOGY, 2024, 卷号: 14, 期号: 18, 页码: 5439-5449
作者:
Xin, Xin
;
Gao, Peng
;
Li, Shenggang
Adobe PDF(1953Kb)
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浏览/下载:308/54
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提交时间:2024/08/23
Carbon dioxide
Catalyst activity
Chemical activation
Density functional theory
Dissociation
Hydrogen
Hydrogenation
II-VI semiconductors
Oxygen
Oxygen vacancies
Catalyst interfaces
Cu catalyst
Cu catalysts
Cu-catalysts
Heterogeneous catalyst
Hydrogen spill overs
Hydrogen spillover
Model catalysts
Structure-activity relationships
]+ catalyst
Structure and biochemical characterization of L-2-hydroxyglutarate dehydrogenase and its role in the pathogenesis of L-2-hydroxyglutaric aciduria
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2024, 卷号: 300, 期号: 1
作者:
Yang, Jun
;
Chen, Xingchen
;
Jin, Shan
;
Ding, Jianping
Adobe PDF(3335Kb)
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收藏
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浏览/下载:389/0
|
提交时间:2024/01/19
Catalyst activity
Mitochondria
2-hydroxyglutaric aciduria
2-oxoglutarate
Biochemical characterization
Catalytic mechanisms
Drosophilla melanogaster
L-2-hydroxyglutarate dehydrogenase
Mitochondrial membranes
Protein crystallography
Structure characterization
Substrate specificity
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