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Recent advances in targeted degradation in the RAS pathway 期刊论文
FUTURE MEDICINAL CHEMISTRY, 2025, 卷号: 17, 期号: 6
作者:  Ge, Zhiming;  Fan, Zisheng;  He, Wei;  Zhou, Guizhen;  Zhou, Yidi
Adobe PDF(2827Kb)  |  收藏  |  浏览/下载:31/2  |  提交时间:2025/03/25
Synthesis of heterocyclic ring-fused analogs of HMG499 as novel degraders of HMG-CoA reductase that lower cholesterol 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 236
作者:  Li, Xing-Zi;  Jiang, Shi-You;  Li, Guo-Qiang;  Jiang, Qian-Ru;  Li, Jue-Wan
Adobe PDF(5589Kb)  |  收藏  |  浏览/下载:641/1  |  提交时间:2022/05/05
Development of a Brigatinib degrader (SIAIS117) as a potential treatment for ALK positive cancer resistance 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 193
作者:  Sun, Ning;  Ren, Chaowei;  Kong, Ying
Adobe PDF(2719Kb)  |  收藏  |  浏览/下载:642/2  |  提交时间:2020/04/23
Proteolysis Targeting Chimeras (PROTACs) of Anaplastic Lymphoma Kinase (ALK) 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 151, 页码: 304-314
作者:  Zhang, Chengwei;  Han, Xiao-Ran;  Yang, Xiaobao;  Jiang, Biao
Adobe PDF(1870Kb)  |  收藏  |  浏览/下载:829/2  |  提交时间:2018/08/09
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