消息
×
loading..
KMS

浏览/检索结果: 共7条,第1-7条 帮助

已选(0)清除 条数/页:   排序方式:
143D, a novel selective KRASG12C inhibitor exhibits potent antitumor activity in preclinical models 期刊论文
ACTA PHARMACOLOGICA SINICA;, 2023
作者:  Xu, Lan-song;  Zheng, Su-xin;  Mei, Liang-he;  Yang, Ke-xin;  Wang, Ya-fang
Adobe PDF(5479Kb)  |  收藏  |  浏览/下载:347/4  |  提交时间:2023/03/24
Discovery of a novel third-generation EGFR inhibitor and identification of a potential combination strategy to overcome resistance 期刊论文
MOLECULAR CANCER, 2020, 卷号: 19, 期号: 1
作者:  Zhang, Tao;  Qu, Rong;  Chan, Shingpan;  Lai, Mengzhen;  Tong, Linjiang
Adobe PDF(2399Kb)  |  收藏  |  浏览/下载:739/248  |  提交时间:2020/06/17
Discovery and biological evaluation of N-(3-(7-((2-methoxy-4-(4-methylpiperazin-1-yl)phenyl)amino)-4-methyl-2-oxo-2H-pyrimido[4,5-d][1,3]oxazin-1(4H)-yl)phenyl)acrylamide as potent Bruton's tyrosine kinase inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 415-422
作者:  Lai, Meng-zhen;  Song, Pei-ran;  Dou, Dou;  Diao, Yan-yan;  Tong, Lin-jiang
Adobe PDF(3317Kb)  |  收藏  |  浏览/下载:412/0  |  提交时间:2020/03/16
Identification of compound D2923 as a novel anti-tumor agent targeting CSF1R 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 11, 页码: 1768-1776
作者:  Liu, Ying-Qiang;  Wang, Ya-Nan
Adobe PDF(4315Kb)  |  收藏  |  浏览/下载:415/0  |  提交时间:2018/11/13
Identification of small molecule inhibitors targeting the SMARCA2 bromodomain from a high-throughput screening assay 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 9, 页码: 1544-1552
作者:  Lu, Tian;  Hu, Jun-chi;  Lu, Wen-chao;  Han, Jie;  Ding, Hong
Adobe PDF(3143Kb)  |  收藏  |  浏览/下载:541/3  |  提交时间:2018/09/09
The plant sesquiterpene lactone parthenolide inhibits Wnt/-catenin signaling by blocking synthesis of the transcriptional regulators TCF4/LEF1 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: 293, 期号: 14, 页码: 5335-5344
作者:  
Adobe PDF(2532Kb)  |  收藏  |  浏览/下载:557/0  |  提交时间:2018/05/10
Computer-Aided Drug Design in Epigenetics 期刊论文
FRONTIERS IN CHEMISTRY, 2018, 卷号: 6
作者:  Lu, Wenchao;  Zhang, Rukang;  Jiang, Hao;  Zhang, Huimin;  Luo, Cheng
Adobe PDF(3286Kb)  |  收藏  |  浏览/下载:1939/584  |  提交时间:2018/04/11
  • 首页
  • 上一页
  • 1
  • 下一页
  • 末页