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Discovery of GPX4 inhibitors through FP-based high-throughput screening 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265
作者:  Cao, Yu;  Wu, Bin;  Xu, Ying;  Wang, Mingchen;  Wu, Xinyu
Adobe PDF(5751Kb)  |  收藏  |  浏览/下载:257/0  |  提交时间:2024/03/04
Distinct kinetic mechanisms of H3K4 methylation catalyzed by MLL3 and MLL4 core complexes 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2021, 卷号: 296
作者:  Zheng, Yongxin;  Huang, Yinping;  Mencius, Jun;  Li, Yanjing;  Zhao, Lijie
Adobe PDF(1642Kb)  |  收藏  |  浏览/下载:259/0  |  提交时间:2021/12/17
The identification of novel small-molecule inhibitors targeting WDR5-MLL1 interaction through fluorescence polarization based high-throughput screening 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 4, 页码: 638-645
作者:  Ye, Xiaoqing;  Zhang, Rukang;  Lian, Fulin;  Zhang, Weiyao;  Lu, Wenchao
Adobe PDF(5234Kb)  |  收藏  |  浏览/下载:476/1  |  提交时间:2019/02/15
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