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Tuning LLMs with Explicit Knowledge 会议论文
ECML PKDD 2025 - EUROPEAN CONFERENCE ON MACHINE LEARNING AND PRINCIPLES AND PRACTICE OF KNOWLEDGE DISCOVERY IN DATABASES
作者:  Han JQ(韩嘉祺);  Li BQ(李秉千);  Gong QY(龚谦益);  Liu YB(刘宇博);  Zhou Y(周熠)
Adobe PDF(2552Kb)  |  收藏  |  浏览/下载:83/10  |  提交时间:2025/03/05
Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8
作者:  Xu, Lei;  Xuyan, Xuyang;  Minmi, Minmin;  Wang, Zhiji;  Shee, Chao
Adobe PDF(1267Kb)  |  收藏  |  浏览/下载:367/0  |  提交时间:2023/07/24
Rational Design and Development of Novel CDK9 Inhibitors for the Treatment of Acute Myeloid Leukemia 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14647-14663
作者:  Han, Xu;  Song, Ning;  Saidahmatov, Abdusaid;  Wang, Peipei;  Wang, Yong
Adobe PDF(5151Kb)  |  收藏  |  浏览/下载:525/0  |  提交时间:2021/11/19
Discovery of thalidomide-based PROTAC small molecules as the highly efficient SHP2 degraders 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 218
作者:  Yang, Xiangbo;  Wang, Zhijia;  Pei, Yuan;  Song, Ning;  Xu, Lei
Adobe PDF(1954Kb)  |  收藏  |  浏览/下载:306/0  |  提交时间:2021/06/04
Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino) pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 173, 页码: 44-62
作者:  Tong, Lexian;  Song, Pinrao;  Jiang, Kailong;  Xu, Lei;  Jin, Tingting
Adobe PDF(1046Kb)  |  收藏  |  浏览/下载:610/12  |  提交时间:2019/06/04
Exploration of novel macrocyclic dipeptide N-benzyl amides as proteasome inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 423-439
作者:  Yu, Jianjun;  Liu, Jieyu;  Li, Daqiang;  Xu, Lei;  Hong, Duidui
Adobe PDF(3236Kb)  |  收藏  |  浏览/下载:455/7  |  提交时间:2019/02/25
Design, synthesis, and biological evaluation of novel phenol ether derivatives as non-covalent proteasome inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 161, 页码: 543-558
作者:  Yu, Jianjun;  Xu, Lei;  Hong, Duidui;  Zhang, Xiaotuan;  Liu, Jieyu
Adobe PDF(1828Kb)  |  收藏  |  浏览/下载:464/1  |  提交时间:2018/12/15
Development of Macrocyclic Peptides Containing Epoxyketone with Oral Availability as Proteasome Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 20, 页码: 9177-9204
作者:  Li, Daqiang;  Zhang, Xiaotuan;  Ma, Xiaodong;  Xu, Lei;  Yu, Jianjun
Adobe PDF(4610Kb)  |  收藏  |  浏览/下载:644/0  |  提交时间:2018/11/15
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