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IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response 期刊论文
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2025, 卷号: 14, 期号: 1
作者:  Yao, Mingyue;  Yan, Wenzhong;  Wang, Yafang;  Zhao, Yu;  Xu, Xiaowei
Adobe PDF(14589Kb)  |  收藏  |  浏览/下载:69/2  |  提交时间:2025/03/03
Discovery of Novel BCL6-Targeting PROTACs with Effective Antitumor Activities against DLBCL in Vitro and in Vivo 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 277
作者:  Dazhao Mi;  Cheng Li(李成);  Yuzhan Li;  Mingyue Yao;  Yan Li
Adobe PDF(7740Kb)  |  收藏  |  浏览/下载:350/13  |  提交时间:2024/09/02
Structure-based design of pan-coronavirus inhibitors targeting host cathepsin L and calpain-1. 期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 页码: 1651-1664
作者:  xiexiong;  Qiaoshuai Lan;  Jinyi Zhao;  Sulin Zhang;  Liu L(刘露)
Adobe PDF(4198Kb)  |  收藏  |  浏览/下载:316/18  |  提交时间:2024/12/02
Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers 期刊论文
ADVANCED SCIENCE, 2024, 卷号: 11, 期号: 41
作者:  
Adobe PDF(9804Kb)  |  收藏  |  浏览/下载:333/2  |  提交时间:2024/09/20
Targeting ST8SIA6-AS1 counteracts KRASG12C inhibitor resistance through abolishing the reciprocal activation of PLK1/c-Myc signaling 期刊论文
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2023
作者:  Yafang Wang;  Mingyue Yao;  Cheng Li (李成);  Kexin Yang
Adobe PDF(16153Kb)  |  收藏  |  浏览/下载:364/5  |  提交时间:2024/09/02
Design and Synthesis of Triazole-Containing HDAC Inhibitors That Induce Antitumor Effects and Immune Response 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2023
作者:  
Adobe PDF(10205Kb)  |  收藏  |  浏览/下载:408/7  |  提交时间:2023/04/10
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors 期刊论文
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1
作者:  Zang, Yi;  Su, Mingbo;  Wang, Qingxing;  Cheng, Xi;  Zhang, Wenru
Adobe PDF(2374Kb)  |  收藏  |  浏览/下载:750/148  |  提交时间:2023/03/10
Confinement effect induced conformation change of one-dimensional phosphorus chains filled in carbon nanotubes 期刊论文
CARBON, 2022, 卷号: 189, 页码: 467-473
作者:  Yao, Fenfa;  Xia, Mingyue;  Zhang, Qing;  Wu, Qiuqin;  Terasaki, Osamu
Adobe PDF(1907Kb)  |  收藏  |  浏览/下载:373/0  |  提交时间:2022/01/10
Identification of Novel Disruptor of Telomeric Silencing 1-like (DOT1L) Inhibitors through Structure-Based Virtual Screening and Biological Assays 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2016, 卷号: 56, 期号: 3, 页码: 527-534
作者:  Chen, Shijie;  Li, Linjuan;  Chen, Yantao;  Hu, Junchi;  Liu, Jingqiu
Adobe PDF(2144Kb)  |  收藏  |  浏览/下载:656/3  |  提交时间:2017/07/04
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