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Dynamic Cap-Mediated Substrate Access and Potent Inhibitor Design of Monkeypox Virus I7L Protease 期刊论文
ADVANCED SCIENCE, 2025
作者:  Su, Haixia;  Wu, Guoqing;  Xiong, Muya;  Wang, Yuhang;  Cao, Junyuan
Adobe PDF(5337Kb)  |  收藏  |  浏览/下载:41/4  |  提交时间:2025/04/09
Potency Prediction of Covalent Inhibitors against SARS-CoV-2 3CL-like Protease and Multiple Mutants by Multiscale Simulations 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2024, 卷号: 64, 期号: 24
作者:  Muya Xiong;  Tianqing Nie;  Zhewen Li;  Meiyi Hu;  Haixia Su
Adobe PDF(7488Kb)  |  收藏  |  浏览/下载:260/5  |  提交时间:2024/12/02
Discovery of Novel Nonpeptidic and Noncovalent Small Molecule 3CLpro Inhibitors as anti-SARS-CoV-2 Drug Candidate 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15
作者:  Jiang, Zhidong;  Feng, Bo;  Chen, Lu;  Nie, Tianqing;  Chen, Shizhao
Adobe PDF(7849Kb)  |  收藏  |  浏览/下载:193/6  |  提交时间:2024/08/14
Soft MicromotorswithSwitchableMotionEnabledby3D-to-3D Shape Reconfiguration 期刊论文
CHEMISRTY OF MATERIALS, 2024, 卷号: 36, 期号: 9, 页码: 4174-4184
作者:  Chen, Xinran;  Wang, Han;  Meng, Xiao;  He, Yisheng;  Jin, Bowen
Adobe PDF(4781Kb)  |  收藏  |  浏览/下载:301/0  |  提交时间:2024/04/23
Discovery and Mechanism Study of SARS-CoV-2 3C-like Protease Inhibitors with a New Reactive Group 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2023
作者:  Ren, Pengxuan;  Li, Hui;  Nie, Tianqing;  Jian, Xiaoqin;  Yu, Changyue
Adobe PDF(10889Kb)  |  收藏  |  浏览/下载:426/9  |  提交时间:2023/09/08
Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8
作者:  Xu, Lei;  Xuyan, Xuyang;  Minmi, Minmin;  Wang, Zhiji;  Shee, Chao
Adobe PDF(1267Kb)  |  收藏  |  浏览/下载:370/0  |  提交时间:2023/07/24
Structural insights into dimerization and activation of the mGlu2-mGlu3 and mGlu2-mGlu4 heterodimers 期刊论文
CELL RESEARCH, 2023
作者:  Wang, Xinwei;  Wang, Mu;  Xu, Tuo;  Feng, Ye;  Shao, Qiang
Adobe PDF(4526Kb)  |  收藏  |  浏览/下载:736/231  |  提交时间:2023/06/26
Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY;, 2023, 卷号: 249
作者:  Ren, Pengxuan;  Yu, Changyue;  Zhang, Ruxue;  Nie, Tianqing;  Hu, Qiaoyu
Adobe PDF(6012Kb)  |  收藏  |  浏览/下载:575/6  |  提交时间:2023/03/24
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors 期刊论文
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1
作者:  Zang, Yi
Adobe PDF(2374Kb)  |  收藏  |  浏览/下载:770/153  |  提交时间:2023/03/10
一种三环类化合物、其制备方法及其应用 专利
申请号:CN202211132254.X,申请日期: 2023-01-03,类型:发明申请,状态:授权
发明人:  白芳;  柳红;  许叶春;  张磊砢;  任鹏璇
Unknown(3830Kb)  |  收藏  |  浏览/下载:837/0  |  提交时间:2023/01/03
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