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Rimota-Gd: Paramagnetic Probe for In Vivo MRI Studies of the Cannabinoid 1 Receptor Distribution in the Mouse Brain 期刊论文
ACS CHEMICAL NEUROSCIENCE, 2024, 卷号: 15, 期号: 23
作者:  Ouyang, Qi;  Zhao, Fei;  Ye, Jingjing;  Xu, Mengyang;  Pu, Suyun
Adobe PDF(5147Kb)  |  收藏  |  浏览/下载:275/7  |  提交时间:2024/12/04
Reflections from Nobel laureates in chemistry 期刊论文
CELL CHEMICAL BIOLOGY, 2024, 卷号: 31, 期号: 8
作者:  Cech, Thomas R.;  Charpentier, Emmanuelle;  Wuthrich, Kurt;  Ciechanover, Aaron;  Lefkowitz, Robert J.
收藏  |  浏览/下载:267/0  |  提交时间:2024/11/19
Fluorine-19 labeling of the tryptophan residues in the G protein-coupled receptor NK1R using the 5-fluoroindole precursor in Pichia pastoris expression 期刊论文
JOURNAL OF BIOMOLECULAR NMR, 2024
作者:  Pan, Benxun;  Guo, Canyong;  Liu, Dongsheng;  Wuthrich, Kurt
Adobe PDF(2252Kb)  |  收藏  |  浏览/下载:364/1  |  提交时间:2024/05/14
Selective polypeptide ligand binding to the extracellular surface of the transmembrane domains of the class B GPCRs GLP-1R and GCGR 期刊论文
ISCIENCE, 2023, 卷号: 26, 期号: 6
作者:  Wang, Huixia;  Hu, Wanhui;  Xu, Tiandan;  Yuan, Ya;  Liu, Dongsheng
Adobe PDF(6452Kb)  |  收藏  |  浏览/下载:512/2  |  提交时间:2023/08/21
Solvent accessibility of a GPCR transmembrane domain probed by in-membrane chemical modification (IMCM) 期刊论文
FEBS LETTERS, 2023
作者:  Dandan Feng;  Guanru Feng;  Yanzhuo Song;  Kurt Wuthrich
Adobe PDF(571Kb)  |  收藏  |  浏览/下载:506/1  |  提交时间:2023/09/22
Two-Dimensional NMR Spectroscopy of the G Protein-Coupled Receptor A2AAR in Lipid Nanodiscs 期刊论文
MOLECULES, 2023
作者:  Canyong Guo;  Lingyun Yang;  Zhijun Liu;  Dongsheng Liu;  Kurt Wüthrich
Adobe PDF(2850Kb)  |  收藏  |  浏览/下载:409/1  |  提交时间:2023/11/04
Adenosine A2AReceptor (A2AAR) Ligand Screening Using the 19F-NMR Probe FPPA 期刊论文
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2023, 卷号: 145, 期号: 28, 页码: 15061-15064
作者:  Zhang, Jinfeng;  Feng, Dandan;  Cheng, Jianjun;  Wüthrich, Kurt
Adobe PDF(1667Kb)  |  收藏  |  浏览/下载:551/3  |  提交时间:2023/07/28
GPCR structural characterization by NMR spectroscopy in solution 期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2022, 卷号: 54, 期号: 9
作者:  Yang, Lingyun;  Liu, Dongsheng;  Wuethrich, Kurt
Adobe PDF(1243Kb)  |  收藏  |  浏览/下载:488/2  |  提交时间:2023/01/16
Dual-acting antitumor agents targeting the A 2A adenosine receptor and histone deacetylases: Design and synthesis of 4-(furan-2-yl)-1H- pyrazolo[3,4-d]pyrimidin-6-amine derivatives 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 5, 期号: 236, 页码: 1-14
作者:  Zhang, Jinfeng;  Luo, Ziwei;  Duan, Wenwen;  Yang, Kexin;  Ling, Lijun
Adobe PDF(2628Kb)  |  收藏  |  浏览/下载:523/2  |  提交时间:2022/06/10
GPCR large-amplitude dynamics by 19F-NMR of aprepitant bound to the neurokinin 1 receptor 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 15
作者:  Pan, Benxun;  Liu, Dongsheng;  Yang, Lingyun;  Wüthrich, Kurt
Adobe PDF(1505Kb)  |  收藏  |  浏览/下载:505/3  |  提交时间:2022/05/17
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