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D-morphinan analogs with favorable pharmacokinetic profiles as dual-acting antidepressants (vol 287, 117349, 2025) 其他
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025-05-05, 卷号: 289
作者:  Ji, Jing;  Hu, Zhengtao;  Zheng, Fuqiang;  Zheng, Jiefang;  Cheng, Jiaxin
收藏  |  浏览/下载:21/0  |  提交时间:2025/04/14
D-morphinan analogs with favorable pharmacokinetic profiles as dual-acting antidepressants 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287
作者:  Ji, Jing;  Hu, Zhengtao;  Zheng, Fuqiang;  Zheng, Jiefang;  Cheng, Jiaxin
Adobe PDF(7212Kb)  |  收藏  |  浏览/下载:59/2  |  提交时间:2025/03/10
Molecular recognition of morphine and fentanyl by the human mu-opioid receptor 期刊论文
CELL, 2022, 卷号: 185, 期号: 23
作者:  Zhuang, Youwen;  Wang, Yue;  He, Bingqing;  He, Xinheng;  Zhou, X. Edward
Adobe PDF(11596Kb)  |  收藏  |  浏览/下载:565/0  |  提交时间:2023/01/16
Identification of pyrogallol as a warhead in design of covalent inhibitors for the SARS-CoV-2 3CL protease 期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1
作者:  Su, Haixia;  Yao, Sheng;  Zhao, Wenfeng;  Zhang, Yumin;  Liu, Jia
Adobe PDF(1519Kb)  |  收藏  |  浏览/下载:1189/312  |  提交时间:2021/07/16
Automated design and optimization of multitarget schizophrenia drug candidates by deep learning 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 204
作者:  Tan, Xiaoqin;  Jiang, Xiangrui;  He, Yang;  Zhong, Feisheng;  Li, Xutong
Adobe PDF(4301Kb)  |  收藏  |  浏览/下载:354/0  |  提交时间:2020/11/24
Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 163, 页码: 281-294
作者:  Xing, Jing;  Zhang, Rukang;  Jiang, Xiangrui;  Hu, Tianwen;  Wang, Xinjun
Adobe PDF(4202Kb)  |  收藏  |  浏览/下载:451/1  |  提交时间:2019/03/04
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