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Deuterium substitution at the intolerable site as a strategy to mitigate the toxicity of camptothecin derivatives 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296
作者:  Yu, Xianqiang;  Sun, Ziyu;  Liu, Jing;  Huangfu, Shangwei;  Cheng, Qi
Adobe PDF(11608Kb)  |  收藏  |  浏览/下载:14/4  |  提交时间:2025/07/07
A kinase mediator of rhizobial symbiosis and immunity in Medicago 期刊论文
NATURE, 2025
作者:  Wang, Dapeng;  Jin, Rui;  Shi, Xiaobao;  Guo, Haoran;  Tan, Xinhang
Adobe PDF(54315Kb)  |  收藏  |  浏览/下载:22/1  |  提交时间:2025/06/23
靶蛋白降解化合物、其抗肿瘤用途、其中间体及其用途 专利
申请号:US18923448,申请日期: 2025-02-27,类型:发明申请,状态:实质审查
发明人:  Xiaobao Yang;  Biao Jiang;  Renhong Sun;  Chaowei Ren;  Ning Sun
Adobe PDF(15448Kb)  |  收藏  |  浏览/下载:125/0  |  提交时间:2025/02/28
Targeted Degradation of SOS1 Exhibits Potent Anticancer Activity and Overcomes Resistance in KRAS-Mutant Tumors and BCR-ABL-Positive Leukemia 期刊论文
CANCER RESEARCH, 2025, 卷号: 85, 期号: 1, 页码: 101-117
作者:  Luo, Ziwei;  Lin, Chencen;  Yu, Chuwei;  Yuan, Changxian;  Wu, Wenyong
Adobe PDF(22554Kb)  |  收藏  |  浏览/下载:220/9  |  提交时间:2025/01/13
Minimizing DNA trapping while maintaining activity inhibition via selective PARP1 degrader 期刊论文
CELL DEATH & DISEASE, 2024, 卷号: 15, 期号: 12
作者:  Chen, Li;  Zou, Yahui;  Sun, Renhong;  Huang, Mei;  Zhu, Xiaotong
Adobe PDF(6267Kb)  |  收藏  |  浏览/下载:338/8  |  提交时间:2024/12/03
Release of a ubiquitin brake activates OsCERK1-triggered immunity in rice 期刊论文
NATURE, 2024, 卷号: 629, 期号: 8014, 页码: 1158-+
作者:  Wang, Gang;  Chen, Xi;  Yu, Chengzhi;  Shi, Xiaobao;  Lan, Wenxian
Adobe PDF(78518Kb)  |  收藏  |  浏览/下载:240/1  |  提交时间:2024/07/22
Structural basis for substrate and antibiotic recognition by Helicobacter pylori isoleucyl-tRNA synthetase 期刊论文
FEBS LETTERS, 2024, 卷号: 598, 期号: 5, 页码: 521-536
作者:  Chen, Xiaobao;  Guo, Yu;  Shi, Jiawen;  Wang, Yilun;  Guo, Xinyi
Adobe PDF(3053Kb)  |  收藏  |  浏览/下载:439/3  |  提交时间:2024/03/04
Development of the nonreceptor tyrosine kinase FER-targeting PROTACs as a potential strategy for antagonizing ovarian cancer cell motility and invasiveness 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2023, 卷号: 299, 期号: 6
作者:  Zhang, Yanchun;  Xiong, Xuexue;  Sun, Renhong;  Zhu, Xiaotong;  Wang, Chen
Adobe PDF(2978Kb)  |  收藏  |  浏览/下载:428/8  |  提交时间:2024/04/12
Development of the non-receptor tyrosine kinase FER-targeting PROTACs as a potential strategy for antagonizing ovarian cancer cell motility and invasiveness 期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2023
作者:  Yanchun Zhang;  Xuexue Xiong;  Renhong Sun;  Xiaotong Zhu;  Chen Wang
Adobe PDF(2707Kb)  |  收藏  |  浏览/下载:359/4  |  提交时间:2023/09/25
Discovery of novel BCR-ABL PROTACs based on the cereblon E3 ligase design, synthesis, and biological evaluation (vol 223, 113645, 2021) 其他
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023-04-05, 卷号: 252
作者:  Liu, Haixia;  Ding, Xinyu;  Liu, Linyi;  Mi, Qianglong;  Zhao, Quanju
Adobe PDF(3283Kb)  |  收藏  |  浏览/下载:429/5  |  提交时间:2023/05/15
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