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Concurrent inhibition of p300/CBP and FLT3 enhances cytotoxicity and overcomes resistance in acute myeloid leukemia 期刊论文
ACTA PHARMACOLOGICA SINICA, 2025, 卷号: 46, 期号: 5, 页码: 1390-1403
作者:  Chen, Yu-jun;  Zhao, Yu;  Yao, Ming-yue;  Wang, Ya-fang;  Ma, Ming
Adobe PDF(6202Kb)  |  收藏  |  浏览/下载:111/8  |  提交时间:2025/02/12
IHCH9033, a novel class I HDAC inhibitor, synergizes with FLT3 inhibitor and rescues quizartinib resistance in FLT3-ITD AML via enhancing DNA damage response 期刊论文
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2025, 卷号: 14, 期号: 1
作者:  Yao, Mingyue;  Yan, Wenzhong;  Wang, Yafang;  Zhao, Yu;  Xu, Xiaowei
Adobe PDF(14589Kb)  |  收藏  |  浏览/下载:104/5  |  提交时间:2025/03/03
Inhibited peroxidase activity of peroxiredoxin 1 by palmitic acid exacerbates nonalcoholic steatohepatitis in male mice 期刊论文
NATURE COMMUNICATIONS, 2025, 卷号: 16, 期号: 1
作者:  Yin, Wen;  Xu, Heng;  Bai, Zhonghao
Adobe PDF(3161Kb)  |  收藏  |  浏览/下载:80/1  |  提交时间:2025/02/12
Targeted Degradation of SOS1 Exhibits Potent Anticancer Activity and Overcomes Resistance in KRAS-Mutant Tumors and BCR-ABL-Positive Leukemia 期刊论文
CANCER RESEARCH, 2025, 卷号: 85, 期号: 1, 页码: 101-117
作者:  Luo, Ziwei;  Lin, Chencen;  Yu, Chuwei;  Yuan, Changxian;  Wu, Wenyong
Adobe PDF(22554Kb)  |  收藏  |  浏览/下载:202/8  |  提交时间:2025/01/13
Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers 期刊论文
ADVANCED SCIENCE, 2024, 卷号: 11, 期号: 41
作者:  Wang, Yafang;  Xu, Lansong;  Ling, Lijun;  Yao, Mingyue;  Shi, Shangxuan
Adobe PDF(9804Kb)  |  收藏  |  浏览/下载:378/3  |  提交时间:2024/09/20
Multi-Wavelength Metasurface Empowered Cryptography for Heightened Security and Improved Fidelity 期刊论文
LASER & PHOTONICS REVIEWS, 2024, 卷号: 18, 期号: 10
作者:  Gu, Zhen;  Liu, Haoyang;  Zhang, Zhengping;  Wang, Xiong;  Zhang, Hualiang
Adobe PDF(2708Kb)  |  收藏  |  浏览/下载:388/2  |  提交时间:2024/05/20
Structural basis of peptide recognition and activation of endothelin receptors 期刊论文
NATURE COMMUNICATIONS;, 2023, 卷号: 14, 期号: 1
作者:  Ji, Yujie;  Duan, Jia;  Yuan, Qingning;  He, Xinheng;  Yang, Gong
Adobe PDF(2001Kb)  |  收藏  |  浏览/下载:1155/288  |  提交时间:2023/03/24
Mechanism of hormone and allosteric agonist mediated activation of follicle stimulating hormone receptor 期刊论文
NATURE COMMUNICATIONS;, 2023, 卷号: 14, 期号: 1
作者:  Duan, Jia;  Xu, Peiyu;  Zhang, Huibing;  Luan, Xiaodong;  Yang, Jiaqi
Adobe PDF(3025Kb)  |  收藏  |  浏览/下载:1184/210  |  提交时间:2023/03/24
Computing the relative binding affinity of ligands based on a pairwise binding comparison network 期刊论文
NATURE COMPUTATIONAL SCIENCE, 2023, 卷号: 3, 期号: 10, 页码: 860-872
作者:  Yu, Jie;  Li, Zhaojun;  Chen, Geng;  Kong, Xiangtai;  Hu, Jie
Adobe PDF(3742Kb)  |  收藏  |  浏览/下载:496/145  |  提交时间:2023/11/10
三唑酰胺类化合物及其制备方法和用途 专利
申请号:CN202211494346.2,申请日期: 2023-09-29,类型:发明申请,状态:实质审查
发明人:  程建军;  谢成英;  蒋华良;  闫文仲
Adobe PDF(5474Kb)  |  收藏  |  浏览/下载:466/0  |  提交时间:2023/09/29
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