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Discovery and biological evaluation of carborane-containing derivatives as TEAD auto palmitoylation inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 121
作者:  Li, Chaofan;  Zhang, Yingshuang;  Zhang, Ziyin;  Zhang, Yirong;  Song, Yuxuan
Adobe PDF(3973Kb)  |  收藏  |  浏览/下载:80/6  |  提交时间:2025/03/18
Fine-tuning phenoxy silyl scaffolds for the development of glutathione-responsive prodrugs and antibody-drug conjugates 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 120
作者:  Wei, Ding;  Wang, Huihui;  Huangfu, Shangwei;  Qi, Cheng;  Jiang, Yuecheng
Adobe PDF(5369Kb)  |  收藏  |  浏览/下载:90/6  |  提交时间:2025/03/03
Discovery of novel benzo[b][1,4]oxazine derivatives as ferroptosis inhibitors 期刊论文
BIOORGANIC CHEMISTRY, 2025, 卷号: 156
作者:  Wan, Bi-Wen;  Liu, Wei;  Xiao, Yijie;  Lv, Lijie;  Li, Xuan
Adobe PDF(6015Kb)  |  收藏  |  浏览/下载:78/2  |  提交时间:2025/02/17
Amiloride Synergizes with EGFR PROTACs and Inhibitors to Overcome Therapeutic Resistance in NSCLC 期刊论文
BIOORGANIC CHEMISTRY, 2025
作者:  Xiaojuan Qu;  Hongyue Ou;  Yifan Wu;  Biao Jiang;  Xiaoling Song
Adobe PDF(3021Kb)  |  收藏  |  浏览/下载:26/6  |  提交时间:2025/05/27
13,14-seco seco withaphysalins from Physalis minima and their inhibitory effects on NLRP3 inflammasome activation 期刊论文
BIOORGANIC CHEMISTRY, 2024, 卷号: 151
作者:  Hu, Bintao;  Peng, Xia;  Tang, Chunping;  Geng, Meiyu;  Yao, Sheng
Adobe PDF(1660Kb)  |  收藏  |  浏览/下载:304/2  |  提交时间:2024/08/14
Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido [2,3- d ]pyrimidin-7-one-based SOS1 inhibitor 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 107
作者:  Wang, Kun;  Zhou, Zehui;  Ma, Xinyi;  Xu, Jiahang;  Xu, Wangyang
Adobe PDF(1940Kb)  |  收藏  |  浏览/下载:260/2  |  提交时间:2024/06/17
Discovery of a first-in-class protein degrader for the c-ros oncogene 1 (ROS1) 期刊论文
BIOORGANIC CHEMISTRY, 2024, 卷号: Volume 150
作者:  Jiawen Yang;  Yifan Wu;  Qiaoliang Zhu;  Yongqi Wei;  Xiaojuan Qu
Adobe PDF(7882Kb)  |  收藏  |  浏览/下载:440/12  |  提交时间:2024/07/10
Crbn-based molecular Glues: Breakthroughs and perspectives 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2024, 卷号: 104
作者:  An, Juzeng;  Zhang, Xiaojun
Adobe PDF(11468Kb)  |  收藏  |  浏览/下载:285/1  |  提交时间:2024/06/11
A gene-encoded aldehyde tag repurposed from RiPP cyclophane-forming pathway 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 101
作者:  Ma, Suze;  Chen, Heng;  Liu, Shuxun;  Huang, Xuedong;  Mo, Tianlu
Adobe PDF(3377Kb)  |  收藏  |  浏览/下载:233/0  |  提交时间:2024/05/14
2-Phenylcyclopropylmethylamine (PCPMA) as a privileged scaffold for central nervous system drug design 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024
作者:  Huiqiong Li;  Jianjun Cheng
Adobe PDF(4235Kb)  |  收藏  |  浏览/下载:357/6  |  提交时间:2024/09/25
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